Lipids and Lipid Derivatives
Medchemexpress LLC Vasopressin, 8-L-ornithine-, acetate (salt) | 914453-98-8 | 99.6% | 1042.19 | 25 MG
Ornipressin acetate is a potent vasoconstrictor, hemostatic, and renal agent. It functions as a vasopressin agonist specific for the V1 receptor. This compound can be used as a local vasoconstrictor, can reverse hypotension associated with combined general/epidural anesthesia, and exhibits antidiuretic activity. Additionally, Ornipressin acetate reduces renal vascular resistance and enhances renal blood flow in renal failure models.
- Potent vasoconstrictor
- Hemostatic agent
- Renal agent
- Vasopressin V1 receptor agonist
- Can be used as a local vasoconstrictor
- Reverses hypotension associated with combined general/epidural anesthesia
- Exhibits antidiuretic activity
- Reduces renal vascular resistance
- Enhances renal blood flow in renal failure models
Medchemexpress LLC Delmitide acetate | 501019-16-5 | 99.2% | 1288.62 g/mol | C59H105N17O11.C2H4O2 | 5 MG
Delmitide acetate is an orally active D-isomer decapeptide with potent anti-inflammatory activity. It inhibits production of TNF-α, IFN-γ, and IL-12, and up-regulates heme oxygenase-1, making it useful for preclinical studies such as ulcerative colitis and cytokine modulation research.
- Orally active d-isomer decapeptide.
- Inhibits pro-inflammatory cytokines, including TNF-α, IFN-γ, and IL-12.
- Up-regulates heme oxygenase-1 to modulate inflammatory response.
- Suitable for ulcerative colitis and inflammation studies.
- Provided as an acetate salt in small research quantities.
- High purity suitable for preclinical research.
Cayman Chemical VItamIn K1 2 3-epoxIde 500ug
The inactive metabolite of vitamin K1 formed during blood clotting that is rapidly reduced back to vitamin K1 by a microsomal epoxide reductase
Medchemexpress LLC Abiraterone acetate (Standard) | 154229-18-2 | 99.8% | C₂₆H₃₃NO₂ | 5 MG
Abiraterone acetate (Standard) is the analytical standard of Abiraterone acetate, intended for research and analytical applications. It is an oral, potent, selective, and irreversible inhibitor of CYP17A1 with antiandrogen activity, and is a proagent form of Abiraterone. This compound is used as a reference standard supplied assay.
- Intended for research and analytical applications
- Used in qualitative research experiments
- Used in quantitative research experiments
- Used in methodological research experiments in HPLC, GC, and MS
Medchemexpress LLC BIMAX2 acetate | 98.7% | 3561.98 | 5 MG
BIMAX2 acetate is a high-affinity nuclear localization signal (NLS) peptide that mimics the activity of the classical nuclear localization signal (cNLS). It competitively binds to importin α, inhibiting the binding of cNLS-cargo proteins to importin α. This peptide is useful for studying the role of RBBP4 in regulating nuclear import efficiency and cell senescence.
- Mimics classical nuclear localization signal (cNLS) activity.
- Competitively binds to importin α.
- Inhibits binding of cNLS-cargo proteins to importin α.
- Useful for studying the role of RBBP4 in regulating nuclear import efficiency and cell senescence.
Medchemexpress LLC NN1213 acetate | 99.65% | 4553.10 (free base) | 25 MG
NN1213 acetate is a long-acting human amylin peptide analog and a selective Amylin receptor agonist. It has shown to significantly reduce food intake and fat mass, and can reduce body weight in diet-induced obese rats. This product is suitable for research related to obesity.
- Long-acting human amylin peptide analog
- Selective amylin receptor agonist
- Reduces food intake and fat mass
- Decreases body weight in diet-induced obese rats
- Used for obesity research
Medchemexpress LLC Macupatide acetate | 99.7% | 4984.60 | 25 MG
Macupatide acetate is a glucose-dependent insulinotropic polypeptide (GIP) receptor agonist. It is used in the research of type 2 diabetes by improving insulin secretion responses and insulin sensitivity. Preclinical studies suggest it reduces body weight and fasting blood glucose.
- Improves insulin secretion responses
- Improves insulin sensitivity
- Produces larger insulin sensitivity improvement compared to selective GLP-1 RA dulaglutide
- Combination therapy with GLP-1 RA dulaglutide had additive effects on insulin sensitivity
- Reduces body weight in patients with type 2 diabetes
- Reduces fasting blood glucose in patients with type 2 diabetes
Medchemexpress LLC Lanreotide (acetate) | 2378114-72-6 | 99.8% | 1156.38 | 5 MG
Lanreotide acetate is a somatostatin analogue with antineoplastic activity, primarily used in research for conditions such as carcinoid syndrome.
- Enhances radiation-induced apoptosis
- Inhibits GH-secreting pituitary adenoma cell proliferation and hormone release in vitro
- Induces tumor growth inhibition in male nude mice
Medchemexpress LLC Seglitide acetate | 99248-33-6 | 99.3% | 869.02 g/mol | C46H60N8O9 | 5 MG
Seglitide acetate is a cyclic peptide somatostatin receptor 2 (SSTR2) agonist used in pharmacology research to study somatostatin receptor signaling and regulation of hormone secretion. Supplied as an acetate salt in solid form, it is typically dissolved in DMSO for in vitro and in vivo experiments probing glucagon and growth hormone modulation.
- Potent SSTR2 agonist activity.
- Cyclic peptide sequence for receptor specificity.
- High purity, 99.3%.
- Available in small milligram quantities for research use.
- Soluble in DMSO for straightforward sample preparation.
Medchemexpress LLC JV-1-36 acetate | 221377-79-3 | 99.93% | 3785.88 (free base) | 5 MG
JV-1-36 acetate is a growth hormone-releasing hormone (GHRH) antagonist that demonstrates antioxidant effects, inhibiting reactive oxygen species in A549 lung cancer cells and reducing cell viability in A549 and Hela cells. It is suitable for in vitro research on GHRH antagonists.
- GHRH antagonist
- Inhibits reactive oxygen species in A549 lung cancer cells
- Reduces cell viability in A549 and Hela cells
- Suitable for in vitro research on GHRH antagonists
- Exerts antioxidant effects
Medchemexpress LLC D-α-Tocopherol acetate | 58-95-7 | MFCD00072042 | 98.3% | 50 G
D-α-Tocopherol acetate can be hydrolyzed to d-alpha-tocopherol (VE) and absorbed in the small intestine. It has been shown to inhibit LPS-induced production of NO, prostaglandin E2, and pro-inflammatory cytokines (TNF-α, IFN-γ, IL-1β, and IL-6) in mouse peritoneal macrophages. Additionally, it exhibits a slight suppression on the activation of NF-κB p50 and p65.
- Can be hydrolyzed to d-alpha-tocopherol (VE) and absorbed in the small intestine.
- Inhibits LPS-induced production of NO, prostaglandin E2, and pro-inflammatory cytokines.
- Slightly suppresses activation of NF-κB p50 and p65.
- For research use only.
Medchemexpress LLC Mdp1 (acetate) | 99.7% | 2521.05 | 25 MG
MDP1 acetate is a Melittin-derived peptide that alters the integrity of both Gram-positive and Gram-negative bacterial membranes, effectively killing bacteria through membrane damage. It demonstrates high-antibacterial activity against multidrug-resistant (MDR) and reference strains of S. aureus, E. coli, and P. aeruginosa.
- Alters the integrity of bacterial membranes
- Effective against gram-positive and gram-negative bacteria
- High-antibacterial activity against multidrug-resistant strains
- Potent against S. aureus, E. coli, and P. aeruginosa
- Exhibits time-dependent antibacterial activity
- Induces vesicle or pore formation and cell lysis in bacteria
Medchemexpress LLC Temporin B (acetate) | 99.0% | 1511.89 | 25 MG
Temporin B acetate is a laboratory chemical primarily used for the manufacture of substances. This product is for research use only and intended for experienced personnel and qualified scientists in authorized facilities. It has not been fully validated for medical applications.
- White to off-white solid appearance
- Purity of 99.0% by HPLC
- Recommended for sealed storage, away from moisture
- Powder is stable for 2 years at -80°C
- Powder is stable for 1 year at -20°C
- In solvent, stable for 6 months at -80°C
- In solvent, stable for 1 month at -20°C
Medchemexpress LLC (rel)-β-Tocopherol | 148-03-8 | 99.9% | 416.69 | 10 MG
(rel)-β-Tocopherol is a relative configuration of β-Tocopherol, a lipid-soluble form of vitamin E. It exhibits antioxidant activity and is utilized in various biological studies.
- Functions as a relative configuration of β-Tocopherol.
- Provides antioxidant activity.
- Slightly inhibits A7r5 and CHO cell proliferation.
- Inhibits PMA-induced adhesion of human erythroleukemia (HEL) cells.
- Inhibits the expression of integrins α4 and α5 on cell surface.